1

Fezolinetant

1. (R)-3-Methylpiperazin-2-one

922178-61-8

2

Ethyl 3-methyl-1,2,4-thiadiazole-5-carboxylate

76162-56-6

3

3-Methyl-1,2,4-thiadiazole-5-carbohydrazide

1375066-73-1

4

(8R)-5,6,7,8-Tetrahydro-8-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1,2,4-triazolo[4,3-a]pyrazine 

1429558-08-6

5

Gefapixant Citrate

4-Bromo-2- (propyl-2-yl) phenol eutectic

26307-50-6

6

5- [[4-methoxy-2- (propyl-2-yl) phenyl] oxy] pyrimidine-2,4-diamine

865304-71-8

7

5- [(2,4-diaminopyrimidin-5-yl) oxy] -2-methoxy-4- (propyl-2-yl) benzenesulfonamide

/

8

Vericiguat

5-fluoro-1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridine-3-carboximidamide hydrochloride

1426309-48-9

9

5-Fluoro-1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridine-3-carbonitrile

1350653-26-7

10

(E)-2-(5-fluoro-1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl)-5-(phenyldiazenyl)pyrimidine-4,6-diamine

1350653-29-0

11

2-(5-fluoro-1-(2-fluorobenzyl)-1H-pyrazolo [3,4-b]pyridin-3-yl)pyrimidine-4,5,6-triamine

1350653-30-3

12

5-fluoro-1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridine-3-carbonitrile

1350653-23-4

13

Osimertinib Mesylate

3-(2-chloropyrimidin-4-yl)-1-methyl-1H-indole

1032452-86-0

14

N-(4-fluoro-2-methoxy-5-nitrophenyl)-4-(1-methyl-1H-indol-3-yl)pyrimidin-2-amine

1421372-94-2

15

N1-(2-(dimethylamino)ethyl)-5-methoxy-N1-methyl-N4-(4-(1-methyl-1H-indol-3-yl)pyrimidin-2-yl)-2-nitrobenzene-1,4-diamine

1421372-67-9

16

Elacestrant HCl

(R)-6-(2-amino-4-methoxyphenyl)-5,6,7,8-tetrahydronaphthalen-2-ol

722520-36-7

17

(R)-N-Ethyl-3-[4-(ethyl(2-(6-hydroxy-1,2,3,4-tetradronaphthalen-2-yl)-5-methoxyphenyl)amino)methyl]propionamide

/

18

Amenamevir

4-(1,2,4-oxadiazol-3-yl)aniline

59908-70-2

19

2H-Thiopyran-4-carboxamide, N-(2,6-dimethylphenyl)tetrahydro-, 1,1-dioxide

1798641-63-0

20

Resmetirom

3,5-Dichloro-4-((6-chloro-5-isopropylpyridazin-3-yl)oxy)aniline

920509-27-9

21

(Z)-ethyl (2-cyano-2-(2-(3,5-dichloro-4-((5-isopropyl-6-oxo-1,6-dihydropyridazin-3-yl)oxy)phenyl)hydrazono)acetyl)carbamate

920509-33-7

22

6-(4-amino-2,6-dichlorophenoxy)-4-isopropylpyridazin-3(2H)-one

920509-28-0

23

Linzagolix choline

5-[(2,3-difluoro-6-methoxyphenyl)methoxy]-2-fluoro-4-methoxyaniline

935287-59-5

24

4-[3-[5-[(2,3-twofluorine-6-methoxyphenyl)methoxy]-2-fluoro-4-methoxyphenyl]ureabase]thiophene-2,3-dimethyl2formicacid

1581731-16-9

25

3-[5-[(2,3-twofluorine-6-methoxyphenyl)methoxy]-2-fluoro-4-methoxyphenyl]-2,4-2-1,2,3,4-tetrahydrothiopheneoxygengenerationand[3,4-d]pyrimidine-5-formicacid

935283-04-8

26

Daridorexant Hydrochloride

(S)-1-[5-methoxy-2-(2H-1,2,3-triazol-2-yl)benzoyl]-2-methylpyrrolidine-2-carboxylicacidmethylester

/

27

(S)-1-[5-methoxy-2-(2H-1,2,3-triazol-2-yl)benzoyl]-2-methylpyrrolidine-2-carboxylicacid

/

28

(S)[2-[[6-[(tertbutoxycarbonyl)amino]-3-chloro-2-methylphenyl]carbamoyl]-2-methylpyrrolidin-1-yl][5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl]ketone

/

29

(S)[2-(5-Chloro-4-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl][5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl]ketone

1505484-82-1

30

Elagolix Sodium

Elagolix Sodium Compound IIIa Benzoate

/

31

1-[[2-Fluoro-6-(trifluoromethyl)phenyl]methyl]-6-methylpyrimidine-2,4(1H,3H)-dione

1150560-54-5

32

(2-Fluoro-3-methoxyphenyl)boronic acid

352303-67-4

33

Ethyl 4-bromobutanoate

2969-81-5

34

1-[[2-Fluoro-6-(trifluoromethyl)phenyl]methyl]-5-iodo-6-methylpyrimidine-2,4(1H,3H)-dione

1150560-54-5

35

5-(2-Fluoro-3-methoxyphenyl)-1-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]-6-methylpyrimidine-2,4(1H,3H)-dione

1150560-59-0

36

Daprodustat

1,3-Dicyclohexylbarbituric acid

35824-91-0

37

Darolutamide

2-chloro-4-(1-(tetrahydro-2H-pyran-2-yl)-1H-pyrazol-5-yl)benzonitrile

1297537-35-9

38

2-chloro-4-(1H-pyrazol-5-yl)benzonitrile

1297537-37-1

39

(S)-4-(1-(2-aminopropyl)-1H-pyrazol-3-yl)-2-chlorobenzonitrile

1297537-41-7

40

(S) -4- [1- (2-aminopropyl) -1H pyrazole-3-yl] -2-chlorobenzonitrile

949034-45-1

41

(S)-5-acetyl-N-(1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-yl)propan-2-yl)-1H-pyrazole-3-carboxamide

1297537-33-7

42

4-Bromo-2-chlorobenzonitrile

154607-01-9

43

1-(Tetrahydro-2H-pyran-2-yl)-1H-pyrazole-5-boronic acid pinacol ester

903550-26-5

44

N-(tert-Butoxycarbonyl)-L-alaninol

79069-13-9

45

N-[(2S)-1-[3-(3-Chloro-4-cyanophenyl)-1H-pyrazol-1-yl]prop-2-yl]-5-acetyl-1H-pyrazole-3-carboxamide

1297538-32-9

46

5-Acetyl-1H-pyrazole-3-carboxylic acid

949034-45-1

47

N-[(2S)-1-[3-(3-Chloro-4-cyanophenyl)-1H-pyrazol-1-yl]prop-2-yl]-5-(1-hydroxyethyl)-1H-pyrazole-3-carboxamide

1297538-32-9

48

Topiroxostat

methyl 2-carbamoylpyridine-4-carboxylate

1379342-46-7

49

methyl 2-cyanoisonicotinate

94413-64-6

50

2-cyanoisonicotinohydrazide

135048-32-7

51

Methyl isonicotinate

2459-09-8

52

4-Cyanopyridine

100-48-1

53

Methyl 2-carbamoylpyridine-4-carboxylate

6937-3-7

54

Methyl 2-cyanopyridine-4-carboxylate

94413-64-6

55

2-Cyanopyridine-4-carboxylic acid hydrazide

/

56

2-Cyanopyridine-4-carboxylic acid (pyridine-4-ylmethyl)hydrazide

/

57

Sorafenib Tosylate

N-Methyl-4-chloro-2-pyridinecarboxamide

220000-87-3

58

p-Aminophenol

123-30-8

59

4-(4-Aminophenoxy)-N-methyl-2-pyridinecarboxamide

284462-37-9

60

4-[4-[3-[4-Chloro-3-(trifluoromethyl)phenyl]ureido]phenoxy]-N2-methylpyridine-2-carboxamide

284461-73-0

61

Relugolix

2-[(2,6-Difluorobenzyl)(isopropoxycarbonyl)amino]-4-[(dimethylamino)methyl]-5-(4-nitrophenyl)thiophene-3-carboxylate ethyl ester

2636079-27-9

62

2-[(2,6-Difluorobenzyl)(isopropoxycarbonyl)amino]-4-[(dimethylamino)methyl]-5-[4-(3-methoxyureido)phenyl]thiophene-3-carboxylate ethyl ester

/

63

6-Methoxypyridazine-3-amine

7252-84-8

64

2-[(2,6-Difluorobenzyl)(isopropoxycarbonyl)amino]-4-[(dimethylamino)methyl]-5-[4-(3-methoxyureido)phenyl]thiophene-3-carboxylic acid

　/

65

(2,6-Difluorobenzyl)[4-[(dimethylamino)methyl]-3-[(6-methoxypyridazin-3-yl)carbamoyl]-5-[4-(3-methoxyureido)phenyl]thiophen-2-yl]carbamate isopropyl ester

　/

66

Prucalopride Succinate

4-Amino-5-chloro-2,3-dihydrobenzofuran-7-carboxylic acid

123654-26-2

67

1-(3-Methoxypropyl)-4-piperidinamine

179474-79-4

68

4-Amino-5-chloro-2,3-dihydro-N-[1-(3-methoxypropyl)-4-piperidinyl]benzofuran-7-carboxamide

179474-81-8

69

4-Amino-5-chloro-2,3-dihydro-N-[1-(3-methoxypropyl)-4-piperidinyl]benzofuran-7-carboxamide succinate

179474-85-2

70

Pazopanib HCl

1H-Indazole-3-ethanamine

6814-68-2

71

Perampanel

N-(2-Chloropyrimidin-4-YL)-N,2,3-trimethyl-2H-indazol-6-amine

444731-75-3

72

2-(Pyridin-2-yl)acetic acid hydrochloride

13115-43-0

73

Vortioxetine Hydrobromide

2-((2,4-DiMethylphenyl)thio)phenylaMine

1019453-85-0

74

1-Iodo-2,4-dimethylbenzene

4214-28-2

75

Bis(2-chloroethyl)amine hydrochloride

821-48-7

76

1-[2-(2,4-Dimethylphenylthio)phenyl]piperazine hydrochloride

960203-28-5